I C 07 D 409/12 Z C 07 D 413/12
A 00 946 552
I C 07 D 409/12 Z A 01 N 043/40
A 01 204 323
I C07D409/12, C 07 D 413/12,
C07D401/14, C 07 D 405/12,
C07D231/12, C 07 D 401/12,
C07D417/14, C 07 D 409/14,
A61K031/501, A 61 P 003/00
A 01 228 067
B 00974857.5
C 09.11.2000 Q En
H 07.08.2002 R En
E 14.07.2004
F 10.11.1999 JP 32031799
10.12.1999 JP 35223799
K FÜNFGLIEDRIGE N-HETEROCYCLEN
MIT HYPOGLYKÄMISCHER UND
HYPOLIPIDEMISCHER WIRKUNG
O Takeda Chemical Industries, Ltd.
1-1 Doshomachi 4-chome, Chuo-ku
Osaka-shi, Osaka 541-0045 (JP)
N MOMOSE, Yu
8-7 Sumiregaoka 2-chome
Takarazuka-shi, Hyogo 665-0847 (JP)
MAEKAWA, Tsuyoshi
2-21, loi 1-chome Ikaruga-cho
Ikoma-gun, Nara 636-0124 (JP)
ODAKA, Hiroyuki
12-12, Katsuragi 2-chome Kita-ku
Kobe-shi Hyogo 651-1223 (JP)
KIMURA, Hiroyuki
2-20-808, Ohamanakamachi 1-cho
Sakai-shi Osaka 590-0975 (JP)
Q PCT/JP 2000/007877 (En)
R WO 2001/038325 31.5.2001
I C 07 D 409/14 Z C 07 D 409/12
A 01 228 067
I C 07 D 411/12 Z C 07 D 413/12
A 00 946 552
I C07D413/12, C 07 D 333/34,
C07D405/12, C 07 D 407/12,
C07D409/12, C 07 D 411/12,
C07D419/12
A 00 946 552
B 97943629.2
C 26.09.1997 Q En
H 06.10.1999 R En
E 07.07.2004
F 27.09.1996 US 721183
K SULFONAMIDE UND IHRE
DERIVATE, DIE DIE AKTIVITÄT DES
ENDOTHELINS MODULIEREN
O ENCYSIVE PHARMACEUTICALS INC.
6700 West Loop South, 4th Floor
Bellaire, TX 77401 (US)
N WU, Chengde
7979 Westheimer Rd.,
1102
Houston, TX 77063 (US)
RAJU, Bore, Gowda
41010 Cornace Terrace
Fremont, California 94539 (US)
WOODARD, Patricia
3422 Creekstone Drive
Sugarland, TX 77479 (US)
KOGAN, Timothy, P.
3422 Creekstone Drive
Sugarland, TX 77479 (US)
BLOK, Natalie
3610 Lake Street
Houston, TX 77098 (US)
Q PCT/US 1997/017402 (En)
R WO 1998/013366 2.4.1998
I C 07 D 413/12 Z C 07 D 265/24
A 01 122 245
I C 07 D 413/12 Z A 01 N 043/40
A 01 204 323
I C 07 D 413/12 Z C 07 D 409/12
A 01 228 067
I C 07 D 417/04 Z C 07 D 471/04
A 01 047 694
I C 07 D 417/12 Z A 01 N 043/40
A 01 204 323
I C 07 D 417/14 Z C 07 D 471/04
A 01 047 694
I C 07 D 417/14 Z C 07 D 409/12
A 01 228 067
I C 07 D 419/12 Z C 07 D 413/12
A 00 946 552
I C07D471/04, A 61 K 031/505,
A61K031/47, C 07 D 405/04,
C07D417/04, C 07 D 405/14,
C07D417/14
A 01 047 694
B 99902522.4
C 08.01.1999 Q En
H 02.11.2000 R En
E 07.07.2004
F 12.01.1998 GB 9800569
K BICYCLISCHE HETEROAROMATISCHE
VERBINDUNGEN ALS PROTEIN
TYROSINE KINASE INHIBITOREN
O GLAXO GROUP LIMITED
Glaxo Wellcome House Berkeley
Avenue
Greenford, Middlesex UB6 ONN
(GB)
N CARTER, Malcolm Clive
care of GlaxoSmithKline plc.
Gunnells Wood Road
Stevenage, Hertfordshire SG1 2NY
(GB)
COCKERILL, George Stuart
care of GlaxoSmithKline plc.
Gunnells Wood Road
Stevenage, Hertfordshire SG1 2NY
(GB)
GUNTRIP, Stephen Barry
care of GlaxoSmithkline plc,
Gunnells Wood Road
Stevenage, Hertfordshire SG1 2NY
(GB)
LACKEY, Karen Elizabeth
SmithKline Beecham Corp. Five
Moore Drive
Research Triangle Park, NC 27709
(US)
SMITH, Kathryn Jane
care of GlaxosmithKline plc.
Gunnells Wood Road
Stevenage, Hertfordshire SG1 2NY
(GB)
Q PCT/EP 1999/000048 (En)
R WO 1999/035146 15.7.1999
I C07D471/04, C 07 D 207/22,
C07B043/04
A 01 212 321
B 00956706.6
C 01.09.2000 Q En
H 12.06.2002 R En
E 07.07.2004
F 03.09.1999 GB 9920919
K ZWISCHENPRODUKTE FÜR DIE
HERSTELLUNG VON NAPHTHYRIDIN-
3-CARBONSÄURE-DERIVATEN
O LG Life Sciences, Ltd.
20, Yoido-dong, Youngdungpo-gu
Seoul 150-721 (KR)
N GRINTER, Trevor John
SmithKline Beecham Pharm., Old
Powder Mills
Near Leigh, Tonbridge, Kent TN11
9AN (GB)
HOWIE, Simon
SmithKline Beecham Pharm., Old
Powder Mills
Near Leigh, Tonbridge, Kent TN11
9AN (GB)
Q PCT/GB 2000/003358 (En)
R WO 2001/017961 15.3.2001
I C07D471/04, C 07 D 207/22,
C07B043/04
A 01 214 321
B 00958776.7
C 01.09.2000 Q En
H 19.06.2002 R En
E 14.07.2004
F 03.09.1999 GB 9920917
K HERSTELLUNGSVERFAHREN FÜR
DERIVATE DER
NAPHTHYRIDIN-3-CARBONSÄURE
O LG Life Sciences, Ltd.
20, Yoido-dong, Youngdungpo-gu
Seoul 150-721 (KR)
N CHO, Sungwook, LG Chem
Investment, Ltd.
Life Science R&D, 104-1
Moonji-dong
Yusong-gu, Taejon 305-380 (KR)
CHOI, Hoon, LG Chem Investment
Ltd.
Life Science R&D, 104-1
Moonji-dong
Yusong-gu, Taejon 305-380 (KR)
HAYLER, John, David GlaxoSmith-
Kline
Old Powder Mills, Leigh
Tonbridge, Kent TN 11 9AN (GB)
Q PCT/GB 2000/003366 (En)
R WO 2001/018002 15.3.2001
I C07D471/04, A 61 K 031/437,
A61P025/00
A 01 235 827
B 00977693.1
C 22.11.2000 Q En
H 04.09.2002 R En
E 07.07.2004
F 23.11.1999 GB 9927687
K IMIDAZOPYRIDINDERIVATE ALS
LIGANDEN FÜR GABA-REZEPTOREN
O MERCK SHARP & DOHME LTD.
Hertford Road
Hoddesdon, Hertfordshire EN11 9BU
(GB)
N CRAWFORTH, James Michael
Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR (GB)
HARRISON, Timothy
Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR (GB)
OWENS, Andrew Pate
Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR (GB)
ROWLEY, Michael
Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR (GB)
TEALL, Martin Richard
Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR (GB)
GOODACRE, Simon Charles
Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR (GB)
HALLETT, David James
Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR (GB)
Q PCT/GB 2000/004451 (En)
R WO 2001/038326 31.5.2001
I C 07 D 471/10 Z C 07 D 211/58
A 01 235 803
I C 07 D 471/14 Z C 07 D 211/58
A 01 235 803
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